VU 0134992

CAS No. 755002-90-5

VU 0134992 ( —— )

Catalog No. M21660 CAS No. 755002-90-5

VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 143 Get Quote
5MG 212 Get Quote
10MG 318 Get Quote
25MG 536 Get Quote
50MG 764 Get Quote
100MG 1053 Get Quote
500MG 2115 Get Quote
1G Get Quote Get Quote

Biological Information

  • Product Name
    VU 0134992
  • Note
    Research use only not for human use.
  • Brief Description
    VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM.
  • Description
    VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM.
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Potassium Channel
  • Recptor
    Kir4.1
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    755002-90-5
  • Formula Weight
    411.38
  • Molecular Formula
    C20H31BrN2O2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(C)c1ccc(OCC(=O)NC2CC(C)(C)NC(C)(C)C2)c(Br)c1
  • Chemical Name
    2-(2-Bromo-4-isopropylphenoxy)-N-(2266-tetramethylpiperidin-4-yl)acetamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Kharade SV et al. Discovery Characterization and Effects on Renal Fluid and Electrolyte Excretion of the Kir4.1 Potassium Channel Pore Blocker VU0134992. Mol Pharmacol. 2018 Aug;94(2):926-937.
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